Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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2,746
Tocris Bioscience™ Zolantidine dimaleate
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CAS: 104076-39-3 Molecular Formula: C30H39N3O9S
| CAS | 104076-39-3 |
|---|---|
| Molecular Formula | C30H39N3O9S |
2,747
Tocris Bioscience™ PD 146176
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CAS: 4079-26-9 Molecular Formula: C15H11NS
| CAS | 4079-26-9 |
|---|---|
| Molecular Formula | C15H11NS |
2,748
Tocris Bioscience™ R 268712
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Potent and selective inhibitor of TGF-βRI
| Inhibitors | R 268712 |
|---|---|
| Product Type | R 268712 |
| Molecular Weight (g/mol) | 363.39 |
| Purity | >98% |
2,749
Tocris Bioscience™ TASP 0390325
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Potent and selective V1B receptor antagonist; orally bioavailable
| Target | Vasopressin Receptor |
|---|---|
| CAS | 1642187-96-9 |
| Product Type | Antagonist |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C25H29ClFN5O4.HCl |
| Formula Weight | 554.44g/mol |
2,750
Tocris Bioscience™ AGI 5198
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Potent and selective inhibitor of mutant isocitrate dehydrogenase 1 (mIDH1)
| Target | Dehydrogenase Inhibitors |
|---|---|
| CAS | 1355326-35-0 |
| Purity | 0.98 |
| Chemical Name or Material | N-[2-(Cyclohexylamino)-1-(2-methylphenyl)-2-oxoethyl]-N-(3-fluorophenyl)-2-methyl-1 H-Imidazole-1-acetamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C27H31FN4O2 |
2,751
Tocris Bioscience™ AIM 100
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CAS: 873305-35-2 Molecular Formula: C23H21N3O2
| CAS | 873305-35-2 |
|---|---|
| Molecular Formula | C23H21N3O2 |
2,752
Tocris Bioscience™ SJF 1521
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Selective EGFR PROTAC™
2,753
Tocris Bioscience™ CYM 5442 hydrochloride
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Selective S1P1 receptor agonist
| Inhibitors | CYM 5442 hydrochloride |
|---|---|
| CAS | 1783987-80-3 |
| Product Type | CYM 5442 hydrochloride |
| Molecular Weight (g/mol) | 445.94 |
| Purity | >98% |
2,754
Tocris Bioscience™ MMG 11
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TLR2 antagonist
| Target | Toll-like Receptor Antagonists |
|---|---|
| CAS | 313254-94-3 |
| Purity | 97% |
| Chemical Name or Material | Ethyl 5-(2-oxo-2-(2,3,4-trihydroxyphenyl)ethyl)furan-2-carboxylate |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C15H14O7 |
2,755
Tocris Bioscience™ SDZ WAG 994
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CAS: 130714-47-5 Molecular Formula: C17H25N5O4
| CAS | 130714-47-5 |
|---|---|
| Molecular Formula | C17H25N5O4 |
2,756
Tocris Bioscience™ XAC
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CAS: 1962928-23-9 Molecular Formula: C21H30Cl2N6O4
| CAS | 1962928-23-9 |
|---|---|
| Molecular Formula | C21H30Cl2N6O4 |
2,757
Tocris Bioscience™ Zoniporide dihydrochloride
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CAS: 241799-10-0 Molecular Formula: C17H18Cl2N6O
| CAS | 241799-10-0 |
|---|---|
| Molecular Formula | C17H18Cl2N6O |
2,758
Tocris Bioscience™ Masitinib
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Potent colony-stimulating factor 1 receptor (CSF-1R) tyroine kinase inhibitor
| Target | CD117/c-kit |
|---|---|
| CAS | 790299-79-5 |
| Purity | 0.98 |
| Chemical Name or Material | 4-[(4-Methyl-1-piperazinyl)methyl]-N-[4-methyl-3-[[4-(3-pyridinyl)-2-thiazolyl]amino]phenyl]benzamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C28H30N6OS |
2,759
Tocris Bioscience™ JNJ 303
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CAS: 878489-28-2 Molecular Formula: C21H29ClN2O4S
| CAS | 878489-28-2 |
|---|---|
| Molecular Formula | C21H29ClN2O4S |
2,760
Tocris Bioscience™ YIL 781 hydrochloride
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Ghrelin receptor (GHS-R1a) antagonist
| CAS | 875258-85-8 |
|---|---|
| Chemical Name or Material | 6-(4-Fluorophenoxy)-2-methyl-3-[[(3S)-1-(1-methylethyl)-3-piperidinyl]methyl]-4(3H)-quinazolinone hydrochloride |
| Recommended Storage | Desiccate at Room Temperature |
| Molecular Formula | C24H28FN3O2.HCl |
| Formula Weight | Observed MW: 445.96 |
| Assay Percent Range | >98% |